Product Name :
Ruboxistaurin mesylate
CAS No.:
192050-59-2
Purity :
99.87%
Shipping:
Room temperature in the continental U.S. Other areas may vary.
Storage :
In solvent: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
SMILES:
O=C1NC(C(C2=CN(C3=CC=CC=C32)CCO[C@H](CN(C)C)CC4)=C1C5=CN4C6=CC=CC=C56)=O.CS(=O)(O)=O
Product Description :
Ruboxistaurin (LY333531) mesylate is an orally active, selective and ATP competitive PKCβ inhibitor with IC50 values of 4.7 and 5.{{(2-Hydroxypropyl)-β-cyclodextrin} medchemexpress|{(2-Hydroxypropyl)-β-cyclodextrin} {Biochemical Assay Reagents}|{(2-Hydroxypropyl)-β-cyclodextrin} Purity & Documentation|{(2-Hydroxypropyl)-β-cyclodextrin} Formula|{(2-Hydroxypropyl)-β-cyclodextrin} supplier|{(2-Hydroxypropyl)-β-cyclodextrin} Autophagy} 9 nM for PKCβI and PKCβII, respectively.{{TMRE} site|{TMRE} {Fluorescent Dye}|{TMRE} Biological Activity|{TMRE} In Vitro|{TMRE} custom synthesis|{TMRE} Autophagy} Ruboxistaurin mesylate can be used for the research of eye disorders, heart failure and diabetes.
Formula:
C29H32N4O6S
Molecular Weight :
564.65
Synonyms:
LY333531 mesylate
Additional Information:
|CAS No. 192050-59-2 ; |Synonyms LY333531 mesylate ; |Formula C29H32N4O6S ; |Molecular Weight 564.PMID:23398362 65 ; |SMILES O=C1NC(C(C2=CN(C3=CC=CC=C32)CCO[C@H](CN(C)C)CC4)=C1C5=CN4C6=CC=CC=C56)=O.CS(=O)(O)=O ; |Target PKC ; |Product Description Ruboxistaurin (LY333531) mesylate is an orally active, selective and ATP competitive PKCβ inhibitor with IC50 values of 4.7 and 5.9 nM for PKCβI and PKCβII, respectively. Ruboxistaurin mesylate can be used for the research of eye disorders, heart failure and diabetes. ; |Format Solid ; |Color Orange to red ; |Purity 99.87% ; |Shipping Room temperature in the continental U.S. Other areas may vary. ; |Storage In solvent: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light) ; |Solubility Overview Soluble in DMSO